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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T71891 | G-573 | ||
G-573 is an allosteric inhibitor of MEK that is both potent and selective. The IC(50) value for pERK inhibition in HCT116 tumours by G-573 was estimated to be 0.406 µM. The IC(50) values for tumour growth inhibition in... | |||
T69700 | BAP2 | ||
BAP2 is a novel inhibitor of protein disulfide isomerase (PDI). | |||
T60390 | PI-55 | 6-(2-hydroxy-3-methylbenzylamino)purine | Others |
PI-55 (6-(2-hydroxy-3-methylbenzylamino)purine) is a cytokinin receptor inhibitor that exhibits structural similarity to 6-benzylaminopurine (BAP). It competitively inhibits BAP binding on the specific Arabidopsis recept... | |||
T15571 | Imrecoxib | BAP-909 | COX |
Imrecoxib (BAP-909) is a novel and selective cyclooxygenase 2 (COX-2) inhibitor (IC50: 18 nM). It also inhibits COX1- activity (IC50: 115 nM). Imrecoxib has an anti-inflammatory effect. |